hSMG-1 inhibitor 11e
CAS No. 1402452-10-1
hSMG-1 inhibitor 11e ( —— )
产品货号. M28042 CAS No. 1402452-10-1
hSMG-1 inhibitor 11e is a potent and selective hSMG-1 kinase inhibitor with an IC50 of 900-fold selectivity over mTOR (IC50 of 45 nM), PI3Kα/γ (IC50s of 61 nM and 92 nM) and CDK1/CDK2 (IC50s of 32 μM and 7.1 μM).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥1887 | 有现货 |
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5MG | ¥3216 | 有现货 |
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10MG | ¥4771 | 有现货 |
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25MG | ¥7655 | 有现货 |
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50MG | ¥10368 | 有现货 |
|
100MG | 获取报价 | 有现货 |
|
200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称hSMG-1 inhibitor 11e
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述hSMG-1 inhibitor 11e is a potent and selective hSMG-1 kinase inhibitor with an IC50 of 900-fold selectivity over mTOR (IC50 of 45 nM), PI3Kα/γ (IC50s of 61 nM and 92 nM) and CDK1/CDK2 (IC50s of 32 μM and 7.1 μM).
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产品描述hSMG-1 inhibitor 11e is a potent and selective hSMG-1 kinase inhibitor with an IC50 of 900-fold selectivity over mTOR (IC50 of 45 nM), PI3Kα/γ (IC50s of 61 nM and 92 nM) and CDK1/CDK2 (IC50s of 32 μM and 7.1 μM).(In Vitro):hSMG-1 inhibitor 11e exhibits an IC50 of 900-fold selectivity over mTOR (IC50 = 45 nM), PI3Kα/γ (IC50 = 61 nM), PI3Kγ (IC50 = 92 nM), CDK1(IC50 = 32 μM) and CDK2 (IC50 = 7.1 μM).
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同义词——
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通路Others
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靶点Other Targets
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受体COX-1;COX-2;Xanthine Oxidase
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研究领域——
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适应症——
化学信息
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CAS Number1402452-10-1
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分子量517.6
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分子式C26H27N7O3S
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纯度>98% (HPLC)
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溶解度——
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SMILESN/A
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Arimboor R, et al. Tetrahydroamentoflavone (THA) from Semecarpus anacardium as a potent inhibitor of xanthine oxidase. J Ethnopharmacol. 2011 Feb 16;133(3):1117-20.
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